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Synthesis and binding properties of deltorphin I analogues containing [R] and [S]-alpha-hydroxymethylnaphtylalanine

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Olma A., Gniadzik A., Lipkowski A. W., Lachwa M.

Acta Biochimica Polonica

2001

tom 48

nr 4

New analogues of deltorphin I (DT I), in which the phenylalanine residue in position 3 is substituted with amphiphilic a,a-disubstituted amino acid enantiomers, (R) and (S)-a-hydroxymethylnaphtylalanine, were synthesized and tested for u and δ opioid receptor affinity and selectivity. Although both analogues have lower affinity to δ receptors than DT I, they both expressed specificity to δ receptors.

Ograniczanie wyników

1 Acta Biochimica Polonica

1 Gniadzik A.

1 Lachwa M.

1 Lipkowski A. W.

1 Olma A.

1 2001

Wyniki wyszukiwania

Synthesis and binding properties of deltorphin I analogues containing [R] and [S]-alpha-hydroxymethylnaphtylalanine